BMS-986242 is more prone to oxidative metabolism and less susceptible to glucuronidation
Co-treatment with both 50 μM BRL 49653 and 10 μM GW-9662 results in statistically lower viable cell numbers after 7 days when compared to treatment with either 50 μM BRL 49653 (P=0
de Alwis DP
Chemical Name: 6-{[(4-chlorophenyl)methyl]sulfanyl}-3-[2-(3
Quassin (hemihydrate) BMS-986242 is more prone toQuassin (Nigakilactone D) is a bioactive triterpenoid from stem bark extract of Quassia amara. Quassin inhibits P. falciparum with an IC50 of 0. 15 M. Quassin possesses reversible antifertility, anti estrogenic and anti plasmodial activity. Product information CAS Number: 76 78 8 Molecular Weight: 388. 45 Formula: C22H28O6 Chemical Name: (3aR, 3a1S, 6aR, 7aS, 8S, 11aS, 11bS) 2, 10 dimethoxy 3, 3a1, 8, 11a tetramethyl 3a, 4, 6a, 7, 7a, 8, 11a, 11b